Adenosine A2a receptor

mammalian protein found in Homo sapiens
rdfs:label
"Adenosine A2a receptor"@en
skos:altLabel "ADORA2A"@en
"adenosine receptor A2a"@en
"adenosine receptor subtype A2a"@en
schema:description
"mammalian protein found in Homo sapiens"@en
schema:dateModified "2026-01-23T21:03:44+00:00"^^xsd:dateTime
schema:version 2457203376
wikibase:identifiers 39
wikibase:sitelinks 0
wikibase:statements 149
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wd:statement/Q21116162-EDA73659-7D25-4391-A110-44FB480CD97E
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wd:statement/Q21116162-F1B3F1E5-5A27-4D2D-8755-C054FCA0C88C
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wd:statement/Q21116162-F7D215CF-2C82-4EBF-B554-7BFF9BAA0159
p:P702 wd:statement/Q21116162-1B0341EC-30C7-4F15-B4E4-B816A6458B91
p:P703 wd:statement/Q21116162-3E40EB16-A083-4AFF-AC32-48E9080A09B1
p:P705 wd:statement/Q21116162-05B842C9-EC98-485B-87DF-2358BC7B0377
wd:statement/Q21116162-3428208A-7F4D-4BF3-AAED-A184B4A20DAA
wd:statement/Q21116162-44C944F9-8E5C-433D-B36F-0336AEFE56B9
wd:statement/Q21116162-520FDDC0-3E0E-4A2F-8166-5CB42E0EA2D0
wd:statement/Q21116162-5ACD3A90-CF48-48DF-81BB-7D6C115CD85C
wd:statement/Q21116162-7E8D44E0-DBA1-4A54-A615-246720D28810
wd:statement/Q21116162-850A7CD0-DEBB-4CF7-ADE5-2E8A959CE899
wd:statement/Q21116162-97A19C94-C3B2-4240-B2B6-D23E80F0BB2B
wd:statement/Q21116162-AE7F09D7-E426-496A-AFB9-B9C8F187BD4E
wd:statement/Q21116162-D35C3A93-D7DC-4881-90AD-6FAE69D97743
wd:statement/Q21116162-D8A11865-DA2B-4F4F-9A9E-E55505EFECFF
wd:statement/Q21116162-DACB7182-95DD-4BEB-A49D-21EAEBCDB131
p:P7260 wd:statement/Q21116162-EEB99CCA-3947-4B22-AC91-4321425CC8CA
p:direct-normalized/P352 <http://purl.uniprot.org/uniprot/P29274>
p:direct-normalized/P637 <http://purl.uniprot.org/refseq/NP_000666>
<http://purl.uniprot.org/refseq/NP_001265426>
<http://purl.uniprot.org/refseq/NP_001265427>
<http://purl.uniprot.org/refseq/NP_001265428>
<http://purl.uniprot.org/refseq/NP_001265429>
p:direct-normalized/P638 <https://rdf.wwpdb.org/pdb/2YDO>
<https://rdf.wwpdb.org/pdb/2YDV>
<https://rdf.wwpdb.org/pdb/3EML>
<https://rdf.wwpdb.org/pdb/3PWH>
<https://rdf.wwpdb.org/pdb/3QAK>
<https://rdf.wwpdb.org/pdb/3REY>
<https://rdf.wwpdb.org/pdb/3RFM>
<https://rdf.wwpdb.org/pdb/3UZA>
<https://rdf.wwpdb.org/pdb/3UZC>
<https://rdf.wwpdb.org/pdb/3VG9>
<https://rdf.wwpdb.org/pdb/3VGA>
<https://rdf.wwpdb.org/pdb/4EIY>
<https://rdf.wwpdb.org/pdb/4UG2>
<https://rdf.wwpdb.org/pdb/4UHR>
<https://rdf.wwpdb.org/pdb/5IU4>
<https://rdf.wwpdb.org/pdb/5IU7>
<https://rdf.wwpdb.org/pdb/5IU8>
<https://rdf.wwpdb.org/pdb/5IUA>
<https://rdf.wwpdb.org/pdb/5IUB>
wdt:P10376 "agricultural-and-biological-sciences/adenosine-a2a-receptor"
wdt:P129 adenosine
galangin
flavone
sakuranetin
theophylline
morin
BAY 60-6583
CCPA
CGS-21680
CGS 15943
8-cyclopentyl-1,3-dipropylxanthine
caffeine
cyclopentyladenosine
sch-442416
UK-432,097
preladenant
Regadenoson
rolofylline
sch-58261
ZM-241385
istradefylline
wdt:P31 protein
wdt:P352 "P29274"
wdt:P361 Adenosine A2A receptor
G protein-coupled recepteishon
GPCR, rhodopsin-like, 7TM, protein family
wdt:P527 GPCR, rhodopsin-like, 7TM
wdt:P637 "NP_000666"
"NP_001265426"
"NP_001265427"
"NP_001265428"
"NP_001265429"
wdt:P638 "2YDO"
"2YDV"
"3EML"
"3PWH"
"3QAK"
"3REY"
"3RFM"
"3UZA"
"3UZC"
"3VG9"
"3VGA"
"4EIY"
"4UG2"
"4UHR"
"5IU4"
"5IU7"
"5IU8"
"5IUA"
"5IUB"
wdt:P680 enzyme binding
identical protein binding
protein heterodimerization activity
signal transducer activity
G protein-coupled receptor activity
G protein-coupled adenosine receptor activity
alpha-actinin binding
protein binding
type 5 metabotropic glutamate receptor binding
wdt:P681 dendrite
integral component of membrane
membrane
Golgi membrane
soma
integral component of plasma membrane
postsynaptic membrane
presynaptic membrane
presynaptic active zone
asymmetric synapse
axon
glutamatergic synapse
integral component of presynaptic membrane
integral component of postsynaptic membrane
plasma membrane
intermediate filament
postsynaptic density
axolemma
endomembrane system
wdt:P682 sensory perception
prepulse inhibition
inhibitory postsynaptic potential
excitatory postsynaptic potential
central nervous system development
positive regulation of synaptic transmission, glutamatergic
positive regulation of long-term synaptic potentiation
apoptotic process
negative regulation of cell population proliferation
negative regulation of cysteine-type endopeptidase activity involved in apoptotic process
regulation of transcription, DNA-templated
locomotory behavior
G protein-coupled receptor signaling pathway
cell-cell signaling
synaptic transmission, dopaminergic
inflammatory response
negative regulation of neuron apoptotic process
positive regulation of glutamate secretion
response to amphetamine
positive regulation of renal sodium excretion
eating behavior
adenylate cyclase-modulating G protein-coupled receptor signaling pathway
blood circulation
regulation of norepinephrine secretion
vasodilation
astrocyte activation
regulation of calcium ion transport
adenylate cyclase-activating G protein-coupled receptor signaling pathway
negative regulation of inflammatory response
protein kinase C-activating G protein-coupled receptor signaling pathway
synaptic transmission, glutamatergic
regulation of mitochondrial membrane potential
membrane depolarization
cellular defense response
negative regulation of locomotion
neuron projection morphogenesis
negative regulation of protein kinase activity
response to caffeine
positive regulation of urine volume
positive regulation of apoptotic signaling pathway
positive regulation of protein secretion
G protein-coupled adenosine receptor signaling pathway
synaptic transmission, cholinergic
cAMP biosynthetic process
response to alkaloid
negative regulation of vascular permeability
positive regulation of synaptic transmission, GABAergic
blood coagulation
phagocytosis
regulation of synaptic vesicle exocytosis
negative regulation of alpha-beta T cell activation
positive regulation of acetylcholine secretion, neurotransmission
positive regulation of circadian sleep/wake cycle, sleep
signal transduction
wdt:P702 ADORA2A
wdt:P703 man
wdt:P705 "ENSP00000336630"
"ENSP00000397071"
"ENSP00000400190"
"ENSP00000404497"
"ENSP00000414802"
"ENSP00000473799"
"ENSP00000474097"
"ENSP00000474895"
"ENSP00000475000"
"ENSP00000480012"
"ENSP00000481552"
"ENSP00000483102"
wdt:P7260 "9.A.14.3.8"
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